SCHEMBL7304097

SCHEMBL7304097

C[C@@H]1CC[C@@H](C(F)(F)F)N1C[C@@H](O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA2B P29275 1/20 0.47
ADORA1 P30542 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.46
CTSB P07858 2/20 0.44
CASP1 P29466 1/20 0.42
CTRB1 P17538 2/20 0.42
SPPL2A Q8TCT8 1/20 0.42
KLK5 Q9Y337 2/20 0.41
CYP3A4 P08684 2/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 1/20 0.40
BACE1 P56817 4/20 0.40
HRH1 P35367 1/20 0.40
CTSL P07711 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309658 1.00 ADORA3 (0.47) ADORA3ADORA2AADORA2BADORA1TRPM8
SCHEMBL7311967 0.89 ADORA3 (0.62) ADORA3ADORA2AADORA2BADORA1CTSB
SCHEMBL9164592 0.89 ADORA3 (0.62) ADORA3ADORA2AADORA2BADORA1CTSB
SCHEMBL9018608 0.82 ADORA3 (0.45) ADORA3ADORA2AADORA2BADORA1TRPM8
SCHEMBL9171812 0.80 ADORA3 (0.43) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL9164719 0.80 ADORA3 (0.43) ADORA3ADORA2AADORA2BADORA1KLK5
SCHEMBL7300465 0.79 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1TRPM8
SCHEMBL5704587 0.75 TRPM8 (0.57) TRPM8CTSBCTRB1ALDH1A1CTSL
SCHEMBL7304137 0.75 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1TRPM8
SCHEMBL7306807 0.75 ADORA3 (0.49) ADORA3ADORA2AADORA2BADORA1TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528242-A2 Trifluoromethyl containing pseudopeptides BAYER AG (DE) 1993-02-24 EP disclosed