SCHEMBL7300982

SCHEMBL7300982

CC(C)(C)OC(=O)CN1CCc2ccc(C(=O)Nc3ccc(C#N)cc3)cc2C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
DRD2 P14416 3/20 0.51
NAMPT P43490 5/20 0.49
ROCK2 O75116 3/20 0.47
PRKAA2 P54646 1/20 0.46
DRD3 P35462 2/20 0.45
ABCB1 P08183 2/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
MEN1 O00255 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KMT2A Q03164 2/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
DRD5 P21918 1/20 0.44
TNF P01375 1/20 0.43
NOD2 Q9HC29 1/20 0.43
NOD1 Q9Y239 1/20 0.43
ITGB3 P05106 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307274 0.86 ITGB3 (0.60) DRD2ABCB1ABCG2MEN1KMT2A
SCHEMBL7298730 0.82 KDM4E (0.54) KDM4EALDH1A1DRD2ROCK2PRKAA2
Hydrochloric Acid SCHEMBL7323352 0.81 KDM4E (0.53) KDM4EALDH1A1DRD2ROCK2PRKAA2
SCHEMBL7300010 0.80 ITGB3 (0.68) ABCB1ABCG2ITGB3ITGA2B
SCHEMBL7306830 0.79 ACACB (0.48) KDM4EALDH1A1DRD2MEN1KMT2A
SCHEMBL7299565 0.79 NR1H2 (0.44) KDM4EALDH1A1DRD2MEN1KMT2A
SCHEMBL7312182 0.79 MCHR1 (0.54) DRD2NAMPTITGB3ITGA2B
SCHEMBL12277410 0.76 NR1H2 (0.43) KDM4EALDH1A1DRD2MEN1KMT2A
SCHEMBL4418240 0.76 S1PR1 (0.56) KDM4EALDH1A1DRD2RAB9AITGB3
SCHEMBL773073 0.75 DRD2 (0.64) KDM4EALDH1A1DRD2DRD3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709370-B1 Bicyclic compounds useful as platelet aggregation inhibitors MITSUI CHEMICALS INC (JP) 1999-01-13 EP disclosed
US-5629321-A FIBRINOGEN ANTAGONIST MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-13 US disclosed
EP-0709370-A1 Bicyclic compounds useful as platelet aggregation inhibitors MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-05-01 EP disclosed