SCHEMBL7306830

SCHEMBL7306830

COC(=O)c1ccc2c(c1)CN(CC(=O)OC(C)(C)C)CC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.48
PRMT5 O14744 2/20 0.44
WDR77 Q9BQA1 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NR1H2 P55055 1/20 0.43
DRD2 P14416 6/20 0.42
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
XIAP P98170 1/20 0.41
BIRC2 Q13490 1/20 0.41
HDAC6 Q9UBN7 2/20 0.41
LMNA P02545 1/20 0.41
THRB P10828 1/20 0.41
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299565 0.88 NR1H2 (0.44) MEN1KMT2ANR1H2DRD2ALDH1A1
SCHEMBL12277410 0.83 NR1H2 (0.43) MEN1KMT2ANR1H2DRD2ALDH1A1
SCHEMBL24192400 0.83 ACACB (0.51) ACACBPRMT5WDR77MEN1KMT2A
SCHEMBL30782330 0.82 DRD2 (0.48) ACACBMEN1KMT2ADRD2HSD17B10
SCHEMBL29341704 0.81 DRD2 (0.42) MEN1KMT2ANR1H2DRD2ALDH1A1
SCHEMBL2014179 0.80 DRD2 (0.56) PRMT5WDR77MEN1KMT2ADRD2
SCHEMBL7307274 0.80 ITGB3 (0.60) MEN1KMT2ADRD2LMNA
SCHEMBL29589913 0.80 NR1H2 (0.67) NR1H2KDM4EMAPTMAPK1HDAC6
SCHEMBL2277894 0.80 NR1H2 (0.67) NR1H2KDM4EMAPTMAPK1HDAC6
SCHEMBL7300982 0.79 KDM4E (0.55) MEN1KMT2ADRD2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709370-B1 Bicyclic compounds useful as platelet aggregation inhibitors MITSUI CHEMICALS INC (JP) 1999-01-13 EP disclosed
US-5629321-A FIBRINOGEN ANTAGONIST MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-13 US disclosed
EP-0709370-A1 Bicyclic compounds useful as platelet aggregation inhibitors MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-05-01 EP disclosed