SCHEMBL7301110

SCHEMBL7301110

N#Cc1ccc(OCCCc2cccnc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP19A1 P11511 2/20 0.55
SERPINE1 P05121 4/20 0.52
CYP2A6 P11509 1/20 0.49
CYP11B2 P19099 3/20 0.48
CYP11B1 P15538 3/20 0.48
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAOB P27338 1/20 0.47
HRH1 P35367 2/20 0.46
NAAA Q02083 1/20 0.46
TBXAS1 P24557 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3154669 0.82 CYP2D6 (0.58) CYP3A4CYP2D6CYP2C9CYP19A1SERPINE1
SCHEMBL7302933 0.81 MAOB (0.66) MAOBNAAA
SCHEMBL8923501 0.80 SCN8A (0.49) CYP3A4CYP2D6CYP2C9CYP19A1SERPINE1
SCHEMBL23291337 0.79 CHRNA7 (0.65) CYP3A4CYP2D6CYP2C9CYP19A1SERPINE1
SCHEMBL30428139 0.79 CHRNA7 (0.65) CYP3A4CYP2D6CYP2C9CYP19A1SERPINE1
SCHEMBL11542731 0.78 TDP1 (0.66) CYP3A4CYP2D6CYP2C9CYP19A1SERPINE1
SCHEMBL7294953 0.77 GAA (0.56) CYP3A4CYP2D6CYP2C9SERPINE1CYP2A6
SCHEMBL6061937 0.76 MAOB (0.64) MAOBNAAA
SCHEMBL3366231 0.76 CA2 (0.59) CYP3A4CYP2D6CYP2C9SERPINE1CYP2A6
SCHEMBL8484229 0.76 ALDH1A1 (0.51) CYP19A1CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0504574-B1 1,2,4-Oxadiazole derivatives having monoamine oxidase B enzyme-inhibitory activity and method for preparing same WAKAMOTO PHARMA CO LTD (JP) 1996-02-28 EP disclosed
US-5356916-A Treating Parkinson*s disease WAKAMOTO PHARMACEUTICAL CO., LTD. (JP) 1994-10-18 US disclosed
EP-0504574-A1 1,2,4-Oxadiazole derivatives having monoamine oxidase B enzyme-inhibitory activity and method for preparing same Wakamoto Pharmaceutical Co., Ltd. (JP) 1992-09-23 EP disclosed