SCHEMBL7301445

SCHEMBL7301445

Cc1cc(C)c(C2CCNCC2)c(C(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.40
CYP2D6 P10635 1/20 0.40
KMT2A Q03164 1/20 0.40
PLAT P00750 2/20 0.39
DHODH Q02127 3/20 0.38
HTR2C P28335 4/20 0.38
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
NOTUM Q6P988 1/20 0.37
P2RY14 Q15391 3/20 0.37
ADRB3 P13945 2/20 0.37
ADRA2B P18089 2/20 0.37
DRD1 P21728 2/20 0.37
DRD5 P21918 2/20 0.37
ADRA1B P35368 2/20 0.37
TMEM97 Q5BJF2 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7301304 0.98 KDM4E (0.44) KDM4EMEN1CYP2D6KMT2APLAT
SCHEMBL5546531 0.81 HTR2C (0.48) MEN1CYP2D6KMT2APLATHTR2C
SCHEMBL7302348 0.79 KDM4E (0.42) KDM4EMEN1KMT2AALDH1A1MAPT
SCHEMBL27536215 0.76 ACMSD (0.46) KDM4EMAPTNOTUMLMNA
SCHEMBL27544733 0.75 HTR2C (0.40) MEN1CYP2D6KMT2APLATHTR2C
SCHEMBL27516462 0.75 ACMSD (0.47) KDM4EKMT2ADHODHMAPTNOTUM
SCHEMBL7273067 0.75 HTR3E (0.45) KDM4EMEN1CYP2D6KMT2AMAPT
SCHEMBL7267112 0.75 HTR3E (0.45) KDM4EMEN1CYP2D6KMT2AMAPT
SCHEMBL27866187 0.73 MAPT (0.45) KDM4EDHODHALDH1A1MAPTNOTUM
SCHEMBL13646142 0.72 ACMSD (0.50) DHODHHTR2CNOTUMP2RY14ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5252570-A Amidino and guanidino derivatives B.I. ITALIA (IT) 1993-10-12 US disclosed
US-5047410-A Indolyl derivatives and their use as 5-HT3, receptor antagonists ISTITUTO DE ANGELI S.P.A. (IT) 1991-09-10 US disclosed
EP-0351385-A2 New amidino and guanidino derivatives BOEHRINGER INGELHEIM ITALIA S.p.A. (IT) 1990-01-17 EP disclosed