SCHEMBL7301505

SCHEMBL7301505

O=[PH](O)OCc1ccc2ccccc2c1.c1ccc(CCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.47
CYP1A2 P05177 2/20 0.45
SLC1A3 P43003 1/20 0.45
SLC1A2 P43004 1/20 0.45
SLC1A1 P43005 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.43
ALOX5 P09917 1/20 0.42
RAB9A P51151 1/20 0.42
FFAR1 O14842 1/20 0.42
SOX18 P35713 1/20 0.42
CYSLTR1 Q9Y271 1/20 0.40
KMT2A Q03164 2/20 0.40
PPARG P37231 2/20 0.40
SLC13A5 Q86YT5 1/20 0.40
GPR52 Q9Y2T5 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
NCOA2 Q15596 1/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16825144 0.92 RAB9A (0.47) CYP1A2SLC1A3SLC1A2SLC1A1MRGPRX4
SCHEMBL7301887 0.87 PLAU (0.49) PLAUCYP1A2FFAR1SOX18SLC13A5
SCHEMBL915503 0.79 RAB9A (0.50) CYP1A2SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL698616 0.78 TSHR (0.48) CYP1A2RAB9AKMT2A
SCHEMBL15961256 0.76 TSHR (0.46) CYP1A2RAB9AKMT2A
Hydrochloric Acid SCHEMBL7385052 0.76 AGXT (0.46) CYP1A2RAB9AKMT2A
SCHEMBL8670812 0.76 PLAU (0.59) PLAUCYP1A2ALOX5SOX18KMT2A
SCHEMBL7295889 0.75 AKR1B1 (0.51) CYP1A2SLC1A3SLC1A2SLC1A1FFAR1
SCHEMBL29255545 0.74 PTGS1 (0.59) CYP1A2ALOX5RAB9AFFAR1
Ethylene Glycol SCHEMBL28921702 0.73 TSHR (0.43) CYP1A2RAB9AKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35886-E ENDOTHELIN-CONVERTING ENZYME INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-01 US disclosed
EP-0518299-B1 Phosphonic acid derivatives, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-08 EP disclosed
US-5330978-A Cardiovascular disorders, hypotensive agents, vasodilation TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-07-19 US disclosed
EP-0518299-A2 Phosphonic acid derivatives, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed