SCHEMBL7301766

SCHEMBL7301766

COc1ccc([S+]([O-])CC(Cc2ccccc2)C(=O)NO)cc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 5/20 0.56
MMP9 P14780 2/20 0.56
MMP13 P45452 2/20 0.56
MMP2 P08253 3/20 0.48
MMP3 P08254 3/20 0.48
PDE4A P27815 3/20 0.48
PDE4B Q07343 3/20 0.48
PDE4C Q08493 3/20 0.48
PDE4D Q08499 3/20 0.48
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46
KMT2A Q03164 1/20 0.44
ADAM17 P78536 1/20 0.43
POLB P06746 1/20 0.43
FPR2 P25090 1/20 0.43
ACE P12821 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300411 0.77 MMP1 (0.67) MMP1MMP9MMP13MMP2MMP3
SCHEMBL7303121 0.76 MMP2 (0.60) MMP1MMP9MMP13MMP2MMP3
SCHEMBL7308337 0.76 MMP9 (0.55) MMP1MMP9MMP13MMP2MMP3
SCHEMBL13103439 0.72 CYP1A2 (0.63)
SCHEMBL6932424 0.72 MMP13 (0.50) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6931491 0.72 MMP1 (1.00) MMP1MMP9MMP13MMP2MMP3
SCHEMBL6177184 0.72 CYP1A2 (0.69) PPARGPPARAKMT2AFPR2
SCHEMBL13103425 0.70 CYP1A2 (0.60) PPARGKMT2A
SCHEMBL7381660 0.70 MMP2 (0.75) MMP1MMP9MMP13MMP2MMP3
SCHEMBL7381656 0.70 MMP2 (0.75) MMP1MMP9MMP13MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1177821-C Matrix metalloprotease inhibitors - 2004-12-01 CN disclosed
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5932595-A ANTIARTHRITIC AGENT; MULTIPLE SCLEROSIS; OSTEOPOROSIS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIULCER AGENT SYNTEX (U.S.A.) INC. (US) 1999-08-03 US disclosed
CN-1160045-A Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 1997-09-24 CN disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed