SCHEMBL7302361

SCHEMBL7302361

N[C@@H](CC(=O)NC(=O)OCc1ccccc1)C(=O)Oc1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.42
SLC1A1 P43005 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
LTA4H P09960 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
CASP1 P29466 1/20 0.39
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11808809 0.86 SLC1A3 (0.42) SLC1A3SLC1A1CA12CA1CA2
SCHEMBL10805172 0.85 SLC1A3 (0.49) SLC1A3SLC1A1CA12CA1CA2
SCHEMBL6447987 0.82 SLC1A1 (0.59) SLC1A3SLC1A1CA12CA1CA2
SCHEMBL7271113 0.82 SLC1A1 (0.59) SLC1A3SLC1A1CA12CA1CA2
SCHEMBL7742857 0.79 L3MBTL1 (0.51) SLC1A3SLC1A1CA12CA1CA2
SCHEMBL7742009 0.79 L3MBTL1 (0.51) SLC1A3SLC1A1CA12CA1CA2
SCHEMBL8990136 0.76 ALPI (0.54) SLC1A3SLC1A1LTA4HALDH1A1
SCHEMBL8990144 0.76 ALPI (0.54) SLC1A3SLC1A1LTA4HALDH1A1
SCHEMBL7302369 0.76 PSMB1 (0.55) CTSLCTSBCTSSCTSKCASP1
SCHEMBL7151534 0.76 SYK (0.50) CA12CA1LTA4HCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583248-A Amino acid derivatives having antiviral activity HOFFMANN-LA ROCHE INC. (US) 1996-12-10 US disclosed
EP-0512343-B1 Amino acid derivatives and their use as anti-viral agents HOFFMANN LA ROCHE (CH) 1995-08-02 EP disclosed
US-5430041-A Amino acid derivatives having antiviral activity HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
EP-0512343-A2 Amino acid derivatives and their use as anti-viral agents F. HOFFMANN-LA ROCHE AG (CH) 1992-11-11 EP disclosed