SCHEMBL7302369

SCHEMBL7302369

NC(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)Oc1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PSMB1 P20618 1/20 0.55
CTSK P43235 8/20 0.51
PSMB8 P28062 1/20 0.48
PSMB5 P28074 1/20 0.48
CTSS P25774 4/20 0.48
CTSL P07711 3/20 0.48
CTSB P07858 2/20 0.48
MME P08473 1/20 0.47
ECE1 P42892 1/20 0.47
CASP1 P29466 3/20 0.47
ALDH1A1 P00352 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7333172 0.86 CTSK (0.59) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL7333168 0.86 CTSK (0.59) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL2066047 0.86 CTSK (0.54) CTSKCTSSCTSLCTSBALDH1A1
SCHEMBL11808814 0.86 PSMB1 (0.53) PSMB1CTSKPSMB8PSMB5CTSS
SCHEMBL7736831 0.85 KYNU (0.60) PSMB1CTSKPSMB8PSMB5CTSS
SCHEMBL5181237 0.85 KYNU (0.60) PSMB1CTSKPSMB8PSMB5CTSS
SCHEMBL7688519 0.85 PSMB1 (0.57) PSMB1CTSKPSMB8PSMB5CTSS
SCHEMBL7728708 0.84 CTSL (0.55) CTSKCTSSCTSLCTSBCASP1
SCHEMBL8078067 0.83 PSMB1 (0.56) PSMB1CTSKPSMB8PSMB5CTSS
SCHEMBL16494690 0.83 SIRT2 (0.53) CTSKCTSSCTSLECE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5583248-A Amino acid derivatives having antiviral activity HOFFMANN-LA ROCHE INC. (US) 1996-12-10 US disclosed
EP-0512343-B1 Amino acid derivatives and their use as anti-viral agents HOFFMANN LA ROCHE (CH) 1995-08-02 EP disclosed
US-5430041-A Amino acid derivatives having antiviral activity HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
EP-0512343-A2 Amino acid derivatives and their use as anti-viral agents F. HOFFMANN-LA ROCHE AG (CH) 1992-11-11 EP disclosed