SCHEMBL7302607

SCHEMBL7302607

Nc1ccccc1Nc1c(O)ccc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.54
MAPK14 Q16539 1/20 0.49
G6PD P11413 1/20 0.45
HCRTR1 O43613 1/20 0.44
PTPN22 Q9Y2R2 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 3/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
LMNA P02545 1/20 0.43
CYP2D6 P10635 1/20 0.43
HSD17B10 Q99714 3/20 0.42
HPGD P15428 2/20 0.42
CYP3A4 P08684 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29061899 0.84 HSD17B10 (0.53) G6PDHCRTR1PTPN22ALDH1A1GAA
SCHEMBL9116508 0.79 GAA (0.55) G6PDALDH1A1GAAKDM4EMAPT
SCHEMBL7862553 0.78 KDM1A (0.55) KDM1AMAPK14ALDH1A1GAAKDM4E
SCHEMBL4593816 0.76 CDC25B (0.61) G6PDKDM4EMEN1KMT2ALMNA
SCHEMBL15382645 0.76 POLB (0.57) G6PDHCRTR1ALDH1A1GAAKDM4E
SCHEMBL10871261 0.75 G6PD (0.54) KDM1AG6PDHCRTR1PTPN22ALDH1A1
SCHEMBL7161381 0.75 MAPT (0.47) KDM1AMAPK14ALDH1A1GAAKDM4E
SCHEMBL819667 0.74 ALDH1A1 (0.59) KDM1AMAPK14ALDH1A1GAAKDM4E
SCHEMBL28872379 0.74 PTPN22 (0.54) G6PDHCRTR1PTPN22ALDH1A1GAA
SCHEMBL7302129 0.74 MEN1 (0.62) ALDH1A1GAAKDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0520200-B1 Imidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1998-02-18 EP disclosed
US-5210091-A Calcium channel blockers used in treatment of central nervous system disorders NEUROSEARCH A/S (DK) 1993-05-11 US disclosed
EP-0520200-A2 Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1992-12-30 EP disclosed