SCHEMBL7302864

SCHEMBL7302864

[CH2]C(C(C(N)=O)c1cccc2ccccc12)C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 1/20 0.42
ALOX5 P09917 1/20 0.41
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
ACP3 P15309 1/20 0.38
AOC3 Q16853 1/20 0.38
HSD17B10 Q99714 1/20 0.37
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
AURKB Q96GD4 1/20 0.37
HPGD P15428 1/20 0.37
HTT P42858 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1665813 0.82 ALDH1A1 (0.55) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL7295452 0.80 ALDH1A1 (0.42) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL6243896 0.76 ALDH1A1 (0.53) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL6444521 0.76 ALOX5 (0.41) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL6447034 0.74 AOC3 (0.42) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL6709448 0.74 UTS2R (0.41) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL6894430 0.73 ALDH1A1 (0.51) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL1285411 0.73 ALDH1A1 (0.51) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL6897764 0.73 ALDH1A1 (0.51) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5
SCHEMBL9560093 0.73 ALDH1A1 (0.51) ALDH1A1CYP2C9CYP2C19CYP1A2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0521827-B1 Pharmacological active hydrazin derivatives and process for their preparation CIBA GEIGY AG (CH) 1996-09-25 EP disclosed
EP-0521827-A1 Pharmacological active hydrazin derivatives and process for their preparation CIBA-GEIGY AG (CH) 1993-01-07 EP disclosed