SCHEMBL7303034

SCHEMBL7303034

N=C(N)Nc1ccc(C(=O)NCCc2ccc(CCC(=O)O)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.54
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
ITGB3 P05106 5/20 0.50
ITGA2B P08514 5/20 0.50
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
NAMPT P43490 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC1 Q13547 1/20 0.48
EPHX2 P34913 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
ST14 Q9Y5Y6 1/20 0.48
ITGB1 P05556 1/20 0.47
ITGAV P06756 1/20 0.47
ITGB5 P18084 1/20 0.47
NPC1 O15118 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303517 0.90 NR1H4 (0.61) NR1H4ITGB3ITGA2BHDAC1EPHX2
Hydrochloric Acid SCHEMBL9264373 0.89 NR1H4 (0.60) NR1H4ITGB3ITGA2BHDAC1EPHX2
SCHEMBL7297516 0.87 ST14 (0.64) NR1H4MEN1KMT2AITGB3ITGA2B
SCHEMBL7303178 0.86 MEN1 (0.52) MEN1KMT2ACA12CA1CA2
SCHEMBL4109710 0.86 FFAR1 (0.53) NR1H4ITGB3ITGA2BCA1CA2
SCHEMBL7379804 0.85 ITGB3 (0.55) KMT2AITGB3ITGA2BNAMPTHDAC2
Hydrochloric Acid SCHEMBL9275424 0.85 MAPT (0.51) MEN1KMT2ACA12CA1CA2
SCHEMBL7295673 0.84 MAPT (0.59) NR1H4MEN1KMT2AITGB3ITGA2B
SCHEMBL24892365 0.81 ST14 (0.55) NR1H4MEN1KMT2ACA12CA1
SCHEMBL8500653 0.80 ITGB3 (0.60) ITGB3ITGA2BHDAC2HDAC1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP claimed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US claimed
US-5399585-A Anitcoagulants, antiinflammatory, antitumor HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
US-5084466-A Anticoagulants, antiinflammatory agents, atheriosclerosis and antitumor agents HOFFMANN-LA ROCHE INC. (US) 1992-01-28 US disclosed