SCHEMBL7297516

SCHEMBL7297516

N=C(N)c1ccc(C(=O)NCCc2ccc(CCC(=O)O)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ST14 Q9Y5Y6 2/20 0.64
ITGB3 P05106 7/20 0.60
ITGA2B P08514 7/20 0.60
F2 P00734 1/20 0.56
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
TPSAB1 Q15661 1/20 0.53
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
EPHX2 P34913 1/20 0.52
NR1H4 Q96RI1 1/20 0.52
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
CYP1A2 P05177 1/20 0.50
GAA P10253 1/20 0.50
CYP2D6 P10635 1/20 0.50
MAPT P10636 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303034 0.87 NR1H4 (0.54) ST14ITGB3ITGA2BCA12CA1
SCHEMBL7380405 0.87 F10 (0.58) ST14ITGB3ITGA2BF2HDAC2
SCHEMBL7118598 0.86 ITGB3 (0.74) ST14ITGB3ITGA2BF2CA1
SCHEMBL7304057 0.86 ITGB3 (0.56) ST14ITGB3ITGA2BF2TPSAB1
Hydrochloric Acid SCHEMBL9271862 0.85 ITGB3 (0.55) ST14ITGB3ITGA2BF2TPSAB1
SCHEMBL7303344 0.85 ST14 (0.59) ST14ITGB3ITGA2BF2CA12
Hydrochloric Acid SCHEMBL9272571 0.84 ST14 (0.58) ST14ITGB3ITGA2BF2CA12
SCHEMBL11470600 0.83 ESRRG (0.68) HDAC2HDAC8HDAC6NPC1RAB9A
SCHEMBL9335737 0.83 TPSAB1 (0.67) ST14ITGB3ITGA2BF2CA1
SCHEMBL7303302 0.83 ITGB3 (0.66) ST14ITGB3ITGA2BF2EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP claimed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US claimed
US-5399585-A Anitcoagulants, antiinflammatory, antitumor HOFFMANN-LA ROCHE INC. (US) 1995-03-21 US disclosed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US disclosed
US-5084466-A Anticoagulants, antiinflammatory agents, atheriosclerosis and antitumor agents HOFFMANN-LA ROCHE INC. (US) 1992-01-28 US disclosed