SCHEMBL7303517

SCHEMBL7303517

N=C(N)Nc1ccc(C(=O)NCc2ccc(CCC(=O)O)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 5/20 0.61
EPHX2 P34913 4/20 0.61
PPARG P37231 1/20 0.56
ITGB3 P05106 5/20 0.54
ITGA2B P08514 5/20 0.54
FFAR1 O14842 6/20 0.48
FFAR4 Q5NUL3 2/20 0.48
ITGB1 P05556 1/20 0.47
ITGAV P06756 1/20 0.47
ITGB5 P18084 1/20 0.47
TPSAB1 Q15661 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9264373 0.99 NR1H4 (0.60) NR1H4EPHX2PPARGITGB3ITGA2B
SCHEMBL7303034 0.90 NR1H4 (0.54) NR1H4EPHX2ITGB3ITGA2BITGB1
SCHEMBL7301840 0.86 EPHX2 (0.48) NR1H4EPHX2HDAC1HDAC6
SCHEMBL4109710 0.86 FFAR1 (0.53) NR1H4EPHX2ITGB3ITGA2BFFAR1
SCHEMBL7450519 0.85 PPARG (0.65) NR1H4EPHX2PPARGITGB3ITGA2B
Hydrochloric Acid SCHEMBL9273383 0.85 NR1H4 (0.47) NR1H4EPHX2HDAC1HDAC6
SCHEMBL17894494 0.85 HDAC1 (0.59) NR1H4EPHX2TPSAB1HDAC1HDAC6
SCHEMBL7294446 0.84 EPHX2 (0.52) NR1H4EPHX2TPSAB1HDAC1HDAC6
SCHEMBL7295665 0.81 EPHX2 (0.63) NR1H4EPHX2ITGB3ITGA2BITGB1
Trifluoroacetic Acid SCHEMBL17894404 0.81 EPHX2 (0.53) NR1H4EPHX2PPARGTPSAB1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP claimed
US-5256812-A Antitumor agents, cardiovascular disorders; having amidino or guandino groups HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US claimed