SCHEMBL7303301

SCHEMBL7303301

N=C(N)c1ccc(CC(=O)NCc2ccc(OCC(=O)O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.56
ITGA2B P08514 4/20 0.56
EPHX2 P34913 1/20 0.53
NR1H4 Q96RI1 1/20 0.53
LMNA P02545 2/20 0.50
NPC1 O15118 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MRGPRX1 Q96LB2 1/20 0.50
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 1/20 0.49
THRB P10828 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HPGD P15428 2/20 0.48
KMT2A Q03164 2/20 0.48
PRSS1 P07477 3/20 0.48
F2 P00734 3/20 0.48
TMPRSS6 Q8IU80 2/20 0.48
PRSS2 P07478 2/20 0.48
PRSS3 P35030 2/20 0.48
ST14 Q9Y5Y6 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303187 1.00 ITGB3 (0.56) ITGB3ITGA2BEPHX2NR1H4LMNA
SCHEMBL7293149 0.88 ITGB3 (0.55) ITGB3ITGA2BEPHX2NR1H4LMNA
SCHEMBL9269532 0.88 MAPT (0.54) ITGB3ITGA2BLMNANPC1SMN1; SMN2
SCHEMBL7302582 0.88 MAPT (0.54) ITGB3ITGA2BLMNANPC1SMN1; SMN2
Acetic Acid SCHEMBL9274305 0.87 NPC1 (0.51) ITGB3ITGA2BLMNANPC1SMN1; SMN2
SCHEMBL5037627 0.87 ITGB3 (0.59) ITGB3ITGA2BEPHX2NR1H4LMNA
Hydrochloric Acid SCHEMBL9273979 0.87 MAPT (0.53) ITGB3ITGA2BLMNANPC1SMN1; SMN2
SCHEMBL7442551 0.86 PRSS1 (0.61) ITGB3ITGA2BEPHX2NR1H4LMNA
SCHEMBL7122825 0.82 ITGB3 (0.75) ITGB3ITGA2BPRSS1F2PRSS2
SCHEMBL11787869 0.81 EPHX2 (0.56) ITGB3ITGA2BEPHX2NR1H4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0381033-B1 Carboxylic-acid and sulphonic-acid amides HOFFMANN LA ROCHE (CH) 1994-03-23 EP claimed