SCHEMBL7303497

SCHEMBL7303497

CCCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)c1c(F)cccc1C(F)(F)F)C(=O)CSCc1ccco1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.35
PSMB1 P20618 1/20 0.35
PSMB5 P28074 1/20 0.35
PSMB2 P49721 1/20 0.35
ITGB1 P05556 1/20 0.35
ALDH1A1 P00352 5/20 0.34
POLB P06746 2/20 0.34
MMP3 P08254 2/20 0.33
MMP9 P14780 2/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MMP1 P03956 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7429981 1.00 ITGA4 (0.35) ITGA4PSMB1PSMB5PSMB2ITGB1
SCHEMBL7306044 0.93 PSMB1 (0.40) PSMB1PSMB5PSMB2ALDH1A1POLB
SCHEMBL7306059 0.93 PSMB1 (0.40) PSMB1PSMB5PSMB2ALDH1A1POLB
SCHEMBL7445133 0.88 MMP3 (0.36) ALDH1A1POLBMMP3MMP9NPC1
SCHEMBL8888226 0.88 MMP3 (0.36) ALDH1A1POLBMMP3MMP9NPC1
SCHEMBL7310680 0.88 MMP3 (0.35) PSMB1PSMB5PSMB2ALDH1A1POLB
SCHEMBL7310695 0.88 MMP3 (0.35) PSMB1PSMB5PSMB2ALDH1A1POLB
SCHEMBL7429973 0.88 ALDH1A1 (0.35) ITGA4ITGB1ALDH1A1POLBNPC1
SCHEMBL7312589 0.88 ALDH1A1 (0.39) PSMB1PSMB5PSMB2ALDH1A1POLB
SCHEMBL7312581 0.88 ALDH1A1 (0.39) PSMB1PSMB5PSMB2ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed