SCHEMBL7303768

SCHEMBL7303768

Cc1ccccc1Oc1nc(Cl)cc(Cl)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.48
TSHR P16473 1/20 0.48
RAB9A P51151 1/20 0.48
ALDH1A1 P00352 3/20 0.48
AR P10275 3/20 0.44
HPGD P15428 2/20 0.43
CYP1A2 P05177 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP2C9 P11712 1/20 0.41
HSP90AA1 P07900 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ACHE P22303 3/20 0.38
BCHE P06276 2/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9858859 0.84 SMN1; SMN2 (0.59) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL24287482 0.81 AR (0.50) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL7294576 0.81 ALDH1A1 (0.55) SMN1; SMN2ALDH1A1HSP90AA1L3MBTL1
SCHEMBL8993442 0.81 MEN1 (0.53) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL22724729 0.76 PAX8 (0.51) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL19484600 0.75 HSP90AA1 (0.51) SMN1; SMN2KMT2ARAB9AALDH1A1HSP90AA1
SCHEMBL28796696 0.73 LMNA (0.55) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL29692562 0.73 LMNA (0.55) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL1415796 0.72 PAX8 (0.47) SMN1; SMN2MEN1KMT2ANPC1TSHR
SCHEMBL1748539 0.72 SMN1; SMN2 (0.55) SMN1; SMN2MEN1KMT2ANPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0526708-B1 Sulfonamide, preparation and use thereof as medicine and intermediate HOFFMANN LA ROCHE (CH) 2000-10-18 EP disclosed
US-5292740-A Sulfonamides HOFFMANN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0526708-A1 Sulfonamide, preparation and use thereof as medicine and intermediate F. HOFFMANN-LA ROCHE AG (CH) 1993-02-10 EP disclosed