SCHEMBL7303980

SCHEMBL7303980

COc1ccc2c(c1)c(=O)[nH]c(=O)n2CCCCN1CC=C(c2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 11/20 0.60
HTR1A P08908 1/20 0.58
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 2/20 0.49
POLB P06746 1/20 0.49
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
CASP1 P29466 1/20 0.48
HBB P68871 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308137 0.93 PARP1 (0.60) PARP1HTR1AKDM4EALDH1A1POLB
SCHEMBL7307836 0.91 PARP1 (0.58) PARP1HTR1AKDM4EGAA
SCHEMBL7308205 0.88 PARP1 (0.64) PARP1HTR1AKDM4EALDH1A1MAPT
SCHEMBL7307656 0.86 PARP1 (0.63) PARP1HTR1AMAPT
SCHEMBL7302855 0.86 PARP1 (0.64) PARP1
SCHEMBL7305161 0.85 PARP1 (0.73) PARP1
Bromide SCHEMBL7309634 0.85 PARP1 (0.62) PARP1HTR1AMAPT
Hydrochloric Acid SCHEMBL7301868 0.85 PARP1 (0.62) PARP1KDM4EGAAMAPT
SCHEMBL7288979 0.83 KDM4E (0.58) PARP1HTR1AKDM4EALDH1A1POLB
SCHEMBL7303316 0.83 PARP1 (0.64) PARP1HTR1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US disclosed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP disclosed