SCHEMBL7304539

SCHEMBL7304539

O=C(OCc1ccccc1)N1CCN(C2CCC(O)(c3ccc(F)cc3)CC2)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
RORC P51449 3/20 0.48
CYP2C19 P33261 1/20 0.48
TMEM97 Q5BJF2 5/20 0.47
SIGMAR1 Q99720 5/20 0.47
HTR1A P08908 2/20 0.47
HRH2 P25021 2/20 0.47
HRH1 P35367 2/20 0.47
HRH3 Q9Y5N1 2/20 0.47
ADRA2C P18825 1/20 0.47
CHRM4 P08173 2/20 0.46
TACR1 P25103 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CHRM5 P08912 1/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696969 0.87 RORC (0.58) SMN1; SMN2NPC1RAB9ARORCCYP2C19
SCHEMBL8192046 0.82 HTR1D (0.68)
SCHEMBL29087277 0.80 RORC (0.61) SMN1; SMN2NPC1RAB9ARORCCYP2C19
SCHEMBL18110614 0.80 RORC (0.54) SMN1; SMN2NPC1RAB9ARORCCYP2C19
SCHEMBL7299616 0.79 HTR1D (0.66)
SCHEMBL31628389 0.78 MEN1 (0.55) SMN1; SMN2NPC1RAB9ACYP2C19TMEM97
SCHEMBL29976408 0.78 SMN1; SMN2 (0.54) SMN1; SMN2NPC1RAB9ACYP2C19TMEM97
SCHEMBL7305125 0.78 CCR1 (0.45) RORCHRH3MEN1KMT2A
SCHEMBL13636153 0.78 SIGMAR1 (0.65) SMN1; SMN2NPC1RAB9ACYP2C19TMEM97
SCHEMBL7556949 0.78 CHRM4 (0.61) SMN1; SMN2NPC1RAB9ACYP2C19SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153611-A AS NON-DOPAMINERGIC ANTIISCHEMIC COMPOUNDS FOR TREATING BRAIN DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2000-11-28 US disclosed
EP-0560669-B1 Piperazinyl-and piperidinyl-cyclohexenes and cyclohexanes BRISTOL MYERS SQUIBB CO (US) 1995-06-14 EP disclosed
EP-0560669-A1 Piperazinyl-and piperidinyl-cyclohexenes and cyclohexanes Bristol-Myers Squibb Company (US) 1993-09-15 EP disclosed