SCHEMBL7304749

SCHEMBL7304749

CC(C)[C@H](N)C(=O)N(C(=O)CCc1ccc(O)cc1)[C@@H](CCCC(N)C(=O)OCc1ccccc1)C(=O)NC(C#N)CC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSC P53634 5/20 0.41
CTSK P43235 11/20 0.35
CTSL P07711 10/20 0.35
CTSS P25774 7/20 0.35
CTSB P07858 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CTSH P09668 1/20 0.35
CYP2D6 P10635 1/20 0.35
LNPEP Q9UIQ6 3/20 0.34
ERAP2 Q6P179 2/20 0.34
ERAP1 Q9NZ08 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303940 0.97 CTSC (0.43) CTSCCTSKCTSLCTSSCTSB
SCHEMBL7275336 0.88 CASP1 (0.41) CTSB
SCHEMBL7304440 0.86 F2 (0.38) CTSCCTSKCTSBCYP1A2CYP3A4
SCHEMBL7304203 0.85 CTSC (0.45) CTSC
SCHEMBL7283568 0.84 CASP1 (0.43) CTSLCTSB
SCHEMBL7416641 0.84 CASP1 (0.34) LNPEPERAP2ERAP1
SCHEMBL7417508 0.81 CASP1 (0.35) CTSLLNPEPERAP2ERAP1
SCHEMBL7301728 0.80 CTSC (0.47) CTSCCTSKCTSLCTSSCYP1A2
SCHEMBL7286570 0.73 CASP1 (0.40) CTSBERAP2ERAP1
SCHEMBL7283411 0.71 CASP1 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0547699-A1 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO. INC. (US) 1993-06-23 EP disclosed