SCHEMBL7304773

SCHEMBL7304773

CC(C)(C)OC(=O)N(OC(C)(C)C)C(=O)C1CC(CSc2ccc(Oc3ccccc3)cc2)CCN1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.33
BTK Q06187 4/20 0.33
KCNH2 Q12809 1/20 0.32
SCN3A Q9NY46 1/20 0.32
MCHR1 Q99705 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CPB2 Q96IY4 1/20 0.30
CYP2D6 P10635 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
NPY5R Q15761 1/20 0.30
CSF1R P07333 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309104 0.92 LTA4H (0.30)
SCHEMBL7312101 0.84 MMP13 (0.44) MMP13ALDH1A1
SCHEMBL7731213 0.67 BTK (0.46) MMP13BTKCPB2
SCHEMBL9543647 0.66 GRIK1 (0.33)
SCHEMBL7307600 0.66 MMP13 (0.46) MMP13
SCHEMBL4310678 0.65 FFAR1 (0.46) ALDH1A1
SCHEMBL4310672 0.65 FFAR1 (0.46) ALDH1A1
SCHEMBL9543675 0.62 ELOVL6 (0.33) MMP13
SCHEMBL5548792 0.62 KDM1A (0.52) BTK
SCHEMBL5545060 0.62 KDM1A (0.52) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5932595-A ANTIARTHRITIC AGENT; MULTIPLE SCLEROSIS; OSTEOPOROSIS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIULCER AGENT SYNTEX (U.S.A.) INC. (US) 1999-08-03 US disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed