SCHEMBL9543647

SCHEMBL9543647

CC(C)(C)OC(=O)N(C(=O)[C@@H]1C[C@H](Sc2ccccc2)CCN1)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 2/20 0.33
GRIA2 P42262 1/20 0.33
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
SCN4A P35499 1/20 0.32
GPR119 Q8TDV5 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
HSD11B1 P28845 1/20 0.30
CARM1 Q86X55 1/20 0.30
PRMT6 Q96LA8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543675 0.78 ELOVL6 (0.33)
SCHEMBL7383722 0.75 L3MBTL1 (0.42) GRIK1GRIA2KDM1AL3MBTL1CARM1
SCHEMBL7383725 0.75 L3MBTL1 (0.42) GRIK1GRIA2KDM1AL3MBTL1CARM1
SCHEMBL9543615 0.74 HRH3 (0.42) GPR119
SCHEMBL7420310 0.73 SCN4A (0.43) SCN4A
SCHEMBL7269435 0.70 CXCR3 (0.40)
SCHEMBL8906865 0.69
SCHEMBL27465020 0.69
SCHEMBL7269372 0.69
SCHEMBL8906632 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993018003-A1 SUBSTITUED PIPECOLINIC ACID DERIVATIVES AS HIV PROTEASE INHIBITORS BIO-MEGA/BOEHRINGER INGELHEIM RESEARCH INC. (CA) 1993-09-16 WO disclosed