SCHEMBL7305191

SCHEMBL7305191

COc1ccc(S(=O)(=O)C(CC(=O)NOC(C)(C)C)Cc2ccccc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 12/20 0.76
MMP2 P08253 12/20 0.76
MMP3 P08254 11/20 0.76
PDE4A P27815 8/20 0.76
PDE4B Q07343 8/20 0.76
PDE4C Q08493 8/20 0.76
PDE4D Q08499 8/20 0.76
MMP13 P45452 3/20 0.58
MMP9 P14780 3/20 0.56
CNR1 P21554 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311602 0.92 MMP1 (0.62) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7308348 0.91 MMP1 (0.62) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7302387 0.90 MMP2 (0.60) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7301418 0.89 PDE4A (0.61) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7301051 0.87 MMP1 (0.57) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7308096 0.87 MMP1 (0.57) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL6824624 0.86 MMP2 (1.00) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7311001 0.84 PDE4A (0.56) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7073256 0.83 MMP2 (0.77) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL7311006 0.83 MMP1 (0.56) MMP1MMP2MMP3PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5932595-A ANTIARTHRITIC AGENT; MULTIPLE SCLEROSIS; OSTEOPOROSIS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIULCER AGENT SYNTEX (U.S.A.) INC. (US) 1999-08-03 US disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed