SCHEMBL7305300

SCHEMBL7305300

COc1ccc(OC)c2c1CC[N]C2

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.43
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
ACHE P22303 1/20 0.34
HTR2C P28335 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301417 0.77 DRD2 (0.47)
SCHEMBL2299447 0.77 DRD2 (0.49)
SCHEMBL9404766 0.76 KDM4E (0.44) KDM4EALDH1A1HPGDACHEHTR2C
SCHEMBL9404907 0.76 KDM4E (0.44) KDM4EALDH1A1HPGDACHE
SCHEMBL833885 0.72 ADRA1A (0.59) ADRA1AKDM4EALDH1A1HPGDGLA
SCHEMBL10969055 0.72 ADRA1A (0.59) ADRA1AKDM4EALDH1A1HPGDGLA
SCHEMBL9573096 0.68 HTR2C (0.45) ADRA1AKDM4EALDH1A1HPGDGLA
SCHEMBL5143947 0.67 KDM4E (0.61) ADRA1AKDM4EALDH1A1HPGDGLA
SCHEMBL18183438 0.67 MAOA (0.51) ADRA1AKDM4EALDH1A1HPGDGLA
SCHEMBL443555 0.67 MAOA (0.50) KDM4EALDH1A1GLAGAAHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0614893-B1 Benzoxazine derivatives, their preparation and their use in therapy SYNTHELABO (FR) 1998-05-27 EP claimed
EP-0666250-B1 Derivatives of N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide having neuroprotective and anti-ischemic properties, their preparation and their use, in therapy SYNTHELABO (FR) 1998-02-11 EP claimed
US-5663183-A CEREBRAL DISORDERS SYNTHELABO (FR) 1997-09-02 US claimed
US-5447928-A Antiischemic agents and nervous system disorders SYNTHELABO (FR) 1995-09-05 US claimed
US-5663183-A CEREBRAL DISORDERS SYNTHELABO (FR) 1997-09-02 US disclosed
US-5663183-A CEREBRAL DISORDERS SYNTHELABO (FR) 1997-09-02 US disclosed
US-5550162-A TREATMENT AND PREVENTION OF CEREBRAL DISORDERS SYNTHELABO (FR) 1996-08-27 US disclosed
US-5550162-A TREATMENT AND PREVENTION OF CEREBRAL DISORDERS SYNTHELABO (FR) 1996-08-27 US disclosed
US-5447928-A Antiischemic agents and nervous system disorders SYNTHELABO (FR) 1995-09-05 US disclosed
US-5447928-A Antiischemic agents and nervous system disorders SYNTHELABO (FR) 1995-09-05 US disclosed
EP-0666250-A1 Derivatives of N-(3-aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphthalene-2-carboxamide having neuroprotective and anti-ischemic properties, their preparation and their use, in therapy SYNTHELABO (FR) 1995-08-09 EP disclosed
EP-0614893-A1 Benzoazine derivatives, their preparation and their use in therapy SYNTHELABO (FR) 1994-09-14 EP disclosed