SCHEMBL7305320

SCHEMBL7305320

CC(C)COC(=O)[C@H](CC(=O)OCc1ccccc1)NC(=O)CCCCNC(=O)c1ccc(C(=N)NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.45
HDAC3 O15379 4/20 0.45
HDAC4 P56524 4/20 0.45
HDAC1 Q13547 4/20 0.45
HDAC7 Q8WUI4 4/20 0.45
HDAC2 Q92769 4/20 0.45
HDAC10 Q969S8 4/20 0.45
HDAC11 Q96DB2 4/20 0.45
HDAC8 Q9BY41 4/20 0.45
HDAC9 Q9UKV0 4/20 0.45
HDAC5 Q9UQL6 4/20 0.45
CAPN1 P07384 1/20 0.43
CAPN2 P17655 1/20 0.43
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
MASP2 O00187 2/20 0.40
HSP90AA1 P07900 1/20 0.40
BMP1 P13497 1/20 0.39
ACE P12821 1/20 0.39
SIRT2 Q8IXJ6 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305875 0.86 ACE (0.49) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL7300054 0.82 L3MBTL1 (0.43) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL9217465 0.82 L3MBTL1 (0.43) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL7331153 0.81 HDAC6 (0.53) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL7297749 0.81 MEN1 (0.50) CAPN1CAPN2ACEMEN1KMT2A
SCHEMBL7305313 0.79 HDAC6 (0.49) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL7300378 0.79 HDAC6 (0.54) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL7299527 0.77 ITGB3 (0.44) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL9221804 0.77 ITGB3 (0.44) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL7328520 0.77 ITGB3 (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed