SCHEMBL7305875

SCHEMBL7305875

N=C(NC(=O)OCc1ccccc1)c1ccc(C(=O)NCCCCC(=O)N[C@@H](CC(=O)OCc2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)OCc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACE P12821 1/20 0.49
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
TACR1 P25103 1/20 0.43
PTGER4 P35408 4/20 0.41
HTT P42858 1/20 0.41
BMP1 P13497 1/20 0.41
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305320 0.86 HDAC6 (0.45) ACEHDAC3HDAC4HDAC1HDAC7
SCHEMBL7331153 0.81 HDAC6 (0.53) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7309615 0.81 MAPT (0.56) ACEPOLBMAPTMAPK1
SCHEMBL7300378 0.80 HDAC6 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9223556 0.80 SMN1; SMN2 (0.43) HDAC2HDAC8HDAC6
SCHEMBL7305313 0.78 HDAC6 (0.49) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9215449 0.78 MAPT (0.45) ACEPOLBMAPTMAPK1
SCHEMBL7300054 0.78 L3MBTL1 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9217465 0.78 L3MBTL1 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8407335 0.77 HTT (0.60) HDAC3HDAC4HDAC1HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed