SCHEMBL7306054

SCHEMBL7306054

Oc1cc(C(F)(F)F)cc2ccccc12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.67
NQO2 P16083 1/20 0.55
TRPM4 Q8TD43 1/20 0.52
CYP1A2 P05177 1/20 0.45
HSD17B1 P14061 2/20 0.44
HSD17B2 P37059 2/20 0.44
P2RX1 P51575 2/20 0.43
P2RX4 Q99571 2/20 0.43
P2RX7 Q99572 2/20 0.43
P2RX3 P56373 1/20 0.43
SLC6A2 P23975 1/20 0.40
P2RY14 Q15391 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
ALOX5 P09917 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
USP2 O75604 1/20 0.38
PAK1 Q13153 1/20 0.38
CNR1 P21554 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304418 0.82 PTPN1 (0.59) PTPN1NQO2TRPM4CYP1A2HSD17B1
SCHEMBL720292 0.80 PTPN1 (0.57) PTPN1NQO2TRPM4CYP1A2HSD17B2
SCHEMBL28996781 0.79 PTPN1 (0.56) PTPN1NQO2TRPM4CYP1A2HSD17B1
SCHEMBL20019498 0.78 PTPN1 (0.56) PTPN1NQO2TRPM4CYP1A2ALDH1A1
SCHEMBL8222699 0.78 HSD17B1 (0.58) PTPN1CYP1A2HSD17B1HSD17B2SLC6A2
SCHEMBL29953443 0.77 MGLL (0.43) PTPN1P2RX1P2RX4P2RX7P2RX3
SCHEMBL7670971 0.76 PTPN1 (0.41) PTPN1CYP1A2P2RX1P2RX4P2RX7
SCHEMBL31036112 0.76 PTPN1 (0.41) PTPN1CYP1A2P2RX1P2RX4P2RX7
SCHEMBL4083639 0.76 ALDH1A1 (0.45) PTPN1P2RX1P2RX4P2RX7P2RX3
SCHEMBL7306047 0.76 PTPN1 (0.45) PTPN1CYP1A2P2RX1P2RX4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006042-A Chemical compounds SMITHKLINE BEECHAM CORP (US) 2007-07-25 CN disclosed
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed