SCHEMBL7306166

SCHEMBL7306166

Nc1cc2ccccc2c([O])c1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
HSD17B10 Q99714 5/20 0.43
HPGD P15428 3/20 0.43
CYP3A4 P08684 2/20 0.43
TSHR P16473 2/20 0.43
KEAP1 Q14145 1/20 0.43
HPRT1 P00492 1/20 0.41
KDM4E B2RXH2 3/20 0.40
POLB P06746 2/20 0.40
HTT P42858 1/20 0.40
RAD52 P43351 1/20 0.40
IDO1 P14902 1/20 0.39
HIF1A Q16665 1/20 0.39
CYP1B1 Q16678 1/20 0.39
HTR2A P28223 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
GLA P06280 2/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29463710 0.79 ALDH1A1 (0.48) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL31281983 0.79 ALDH1A1 (0.48) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL677653 0.79 ALDH1A1 (0.48) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL12124161 0.77 ALDH1A1 (0.46) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL7303415 0.77 NSD2 (0.40) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL82369 0.76 ALDH1A1 (0.52) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL3673336 0.74 ALDH1A1 (0.43) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL3668935 0.74 CYP2A6 (0.45) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL7128617 0.74 PTPN22 (0.45) ALDH1A1HSD17B10HPGDCYP3A4TSHR
SCHEMBL3669260 0.74 ALDH1A1 (0.43) ALDH1A1HSD17B10HPGDCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed