SCHEMBL7306293

SCHEMBL7306293

CC(C)C(C#N)(c1ccccc1)S(=O)(=O)CCCC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TBXA2R P21731 2/20 0.36
CYP2D6 P10635 2/20 0.35
CYP1A2 P05177 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC4 P56524 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34
HDAC2 Q92769 2/20 0.34
HDAC10 Q969S8 2/20 0.34
HDAC11 Q96DB2 2/20 0.34
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
HDAC9 Q9UKV0 2/20 0.34
HDAC5 Q9UQL6 2/20 0.34
MAPK1 P28482 1/20 0.34
ADRA1A P35348 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304444 0.82 CYP2D6 (0.34) CYP2C19CYP2D6CYP3A4EBPSIGMAR1
SCHEMBL7316269 0.82 CHRM3 (0.36) CYP2C19ALDH1A1CYP2D6CYP3A4EBP
SCHEMBL7306091 0.71 EBP (0.54) CYP2C19HIF1ATBXA2RCYP2D6CYP1A2
SCHEMBL7304642 0.71 EBP (0.54) CYP2C19HIF1ATBXA2RCYP2D6CYP1A2
SCHEMBL7314859 0.70 TBXA2R (0.35) CYP2C19HIF1AALDH1A1TBXA2RCYP2D6
SCHEMBL7314866 0.69 CES2 (0.35) ALDH1A1TBXA2RHDAC3HDAC4HDAC1
SCHEMBL5751980 0.69 EBP (0.51) CYP2C19HIF1AALDH1A1CYP2D6CYP1A2
SCHEMBL7316961 0.68 ALDH1A1 (0.38) CYP2C19HIF1AALDH1A1TBXA2RCYP2D6
SCHEMBL7309897 0.68 TBXA2R (0.41) CYP2C19ALDH1A1TBXA2RCYP2D6CYP1A2
SCHEMBL7308232 0.66 CYP2C19 (0.39) CYP2C19HIF1AALDH1A1TBXA2RCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed