SCHEMBL7314859

SCHEMBL7314859

CC(C)S(=O)(=O)C(C#N)(CCCCC(=O)O)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35
MAPT P10636 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
CDC25A P30304 2/20 0.34
CDC25B P30305 2/20 0.34
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316961 0.85 ALDH1A1 (0.38) TBXA2RALDH1A1HDAC3HDAC4HDAC1
SCHEMBL7314866 0.81 CES2 (0.35) TBXA2RALDH1A1HDAC3HDAC4HDAC1
SCHEMBL7306130 0.77 CYP2D6 (0.35) CYP3A4CYP2D6SLC22A2SLC22A1PGR
SCHEMBL7304642 0.76 EBP (0.54) TBXA2RHDAC3HDAC4HDAC1HDAC7
SCHEMBL7306091 0.76 EBP (0.54) TBXA2RHDAC3HDAC4HDAC1HDAC7
SCHEMBL7309897 0.74 TBXA2R (0.41) TBXA2RALDH1A1HDAC3HDAC4HDAC1
SCHEMBL7316944 0.72 MEN1 (0.37) SMN1; SMN2
SCHEMBL7308232 0.70 CYP2C19 (0.39) TBXA2RALDH1A1HDAC3HDAC4HDAC1
SCHEMBL7306293 0.70 CYP2C19 (0.36) TBXA2RALDH1A1HDAC3HDAC4HDAC1
SCHEMBL7314215 0.69 SMN1; SMN2 (0.34) TBXA2RALDH1A1CYP3A4SMN1; SMN2SLC22A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed