SCHEMBL7306359

SCHEMBL7306359

N=C(NC(=O)OCc1ccccc1)c1ccc(C(=O)NCCC(=O)NCCC(=O)OCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.46
CTSG P08311 1/20 0.46
CTRB1 P17538 1/20 0.46
CMA1 P23946 1/20 0.46
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
HTT P42858 1/20 0.43
HRH4 Q9H3N8 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7305313 0.95 HDAC6 (0.49) PRSS1CTSGCTRB1CMA1HDAC3
SCHEMBL7331153 0.94 HDAC6 (0.53) PRSS1CTSGCTRB1CMA1HDAC3
SCHEMBL9335659 0.90 HDAC1 (0.48) PRSS1CTSGCTRB1CMA1HDAC3
SCHEMBL9339505 0.87 PPARG (0.47) PRSS1CTSGCTRB1CMA1HDAC2
SCHEMBL7300378 0.86 HDAC6 (0.54) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9222240 0.86 ACE (0.47) HDAC3HDAC1HDAC2MEN1KMT2A
SCHEMBL9217465 0.86 L3MBTL1 (0.43) PRSS1CTSGCTRB1CMA1HDAC3
SCHEMBL7300054 0.86 L3MBTL1 (0.43) PRSS1CTSGCTRB1CMA1HDAC3
SCHEMBL7296073 0.85 ITGB3 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7302006 0.85 SYK (0.46) PRSS1CTSGCTRB1CMA1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed