SCHEMBL7308256

SCHEMBL7308256

CCOC(=O)CC(C(=O)OCC)N1CCN(CC2CN(CC3CCN(CC)CC3)C(=O)O2)CC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
LMNA P02545 1/20 0.38
HTR2B P41595 6/20 0.36
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HRH1 P35367 2/20 0.31
CCR3 P51677 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858160 0.93 ITGB3 (0.34) ITGB3ITGA2BLMNAHTR2BCYP2D6
SCHEMBL7307990 0.90 HTR2B (0.37) ITGB3ITGA2BLMNAHTR2BCYP2D6
SCHEMBL7311057 0.89 ITGB3 (0.40) ITGB3ITGA2BLMNAHTR2BCYP2D6
SCHEMBL7314824 0.88 LMNA (0.42) ITGB3ITGA2BLMNAHTR2B
SCHEMBL7315163 0.87 ITGB3 (0.38) ITGB3ITGA2BHTR2BCYP2D6MAPT
SCHEMBL7304200 0.84 ITGB3 (0.36) ITGB3ITGA2BLMNAHTR2BCYP2D6
SCHEMBL8858185 0.84 ITGB3 (0.33) ITGB3ITGA2BLMNAHTR2B
SCHEMBL7313564 0.83 ITGB3 (0.39) ITGB3ITGA2BLMNAHTR2BCYP2D6
SCHEMBL8858154 0.82 LMNA (0.38) ITGB3ITGA2BLMNAHTR2B
SCHEMBL7303852 0.82 ITGB3 (0.38) ITGB3ITGA2BLMNAHTR2BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed