SCHEMBL7306996

SCHEMBL7306996

CCOC(=O)CC(C(=O)OCC)N1CCN(CC2CN(CCCC3CCN(C(=N)N)CC3)C(=O)O2)CC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
LMNA P02545 1/20 0.34
CYP2D6 P10635 1/20 0.32
KCNH2 Q12809 1/20 0.32
HTR2B P41595 2/20 0.32
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
DRD3 P35462 1/20 0.31
GAA P10253 1/20 0.30
TPSAB1 Q15661 1/20 0.30
TPSD1 Q9BZJ3 1/20 0.30
TPSG1 Q9NRR2 1/20 0.30
PKM P14618 1/20 0.30
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307328 0.98 ITGB3 (0.37) ITGB3ITGA2BLMNACYP2D6KCNH2
SCHEMBL7303852 0.95 ITGB3 (0.38) ITGB3ITGA2BLMNACYP2D6KCNH2
SCHEMBL7311057 0.91 ITGB3 (0.40) ITGB3ITGA2BLMNACYP2D6KCNH2
SCHEMBL7303634 0.90 ITGB3 (0.39) ITGB3ITGA2BCYP2D6HTR2BGAA
SCHEMBL7315964 0.88 ITGB3 (0.40) ITGB3ITGA2BCYP2D6HTR2B
SCHEMBL7303222 0.85 ITGB3 (0.32) ITGB3ITGA2BLMNA
SCHEMBL7309081 0.85 ACHE (0.42) LMNAHTR2B
SCHEMBL7304200 0.84 ITGB3 (0.36) ITGB3ITGA2BLMNACYP2D6HTR2B
SCHEMBL7304230 0.83 HTR2B (0.43) ITGB3ITGA2BLMNACYP2D6HTR2B
SCHEMBL7315730 0.83 ITGB3 (0.33) ITGB3ITGA2BLMNAHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5627197-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-05-06 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed