SCHEMBL7307561

SCHEMBL7307561

CCOC(=O)[C@H](NC(=O)[C@H]1CCCN1C(=O)CCCC[C@@](C#N)(c1ccccc1)C(C)C)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACE P12821 7/20 0.38
ACE2 Q9BYF1 4/20 0.38
F2 P00734 4/20 0.38
CACNA1B Q00975 1/20 0.38
KCNH2 Q12809 1/20 0.37
ELANE P08246 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37
P2RY12 Q9H244 1/20 0.37
PRSS1 P07477 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CMA1 P23946 1/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8083547 0.88 TACR1 (0.44) ACEF2PRSS1DPP4
SCHEMBL7309074 0.88 ACE (0.41) ACEACE2F2PRSS1DPP4
SCHEMBL7309067 0.88 ACE (0.41) ACEACE2F2PRSS1DPP4
SCHEMBL7308379 0.88 TACR1 (0.44) ACEF2PRSS1DPP4
SCHEMBL7308390 0.88 TACR1 (0.44) ACEF2PRSS1DPP4
SCHEMBL7308426 0.88 ACE (0.46) ACEACE2LMNA
SCHEMBL7308435 0.88 ACE (0.46) ACEACE2LMNA
SCHEMBL7316690 0.83 F2 (0.42) ACEF2KMT2APRSS1DPP4
SCHEMBL7316700 0.83 F2 (0.42) ACEF2KMT2APRSS1DPP4
SCHEMBL7306120 0.82 ACE (0.48) ACEACE2DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed