SCHEMBL7307810

SCHEMBL7307810

CC(C)[C@H](NC(=O)N(C)Cc1nc2ccccc2[nH]1)C(=O)Oc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.49
MAPT P10636 9/20 0.48
NPC1 O15118 5/20 0.48
ALDH1A1 P00352 5/20 0.48
RAB9A P51151 4/20 0.48
TDP1 Q9NUW8 4/20 0.48
KDM4E B2RXH2 3/20 0.48
L3MBTL1 Q9Y468 1/20 0.46
SMN1; SMN2 Q16637 5/20 0.45
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
GAA P10253 2/20 0.45
LMNA P02545 2/20 0.44
HTT P42858 1/20 0.44
MAPK1 P28482 3/20 0.43
POLB P06746 1/20 0.43
THRB P10828 1/20 0.42
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
MMP2 P08253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307803 1.00 PKM (0.49) PKMMAPTNPC1ALDH1A1RAB9A
SCHEMBL7302472 0.83 ALDH1A1 (0.50) PKMMAPTNPC1ALDH1A1RAB9A
SCHEMBL7302465 0.83 ALDH1A1 (0.50) PKMMAPTNPC1ALDH1A1RAB9A
SCHEMBL4680503 0.79 CA2 (0.51) MAPTNPC1ALDH1A1RAB9ATDP1
SCHEMBL4680500 0.79 CA2 (0.51) MAPTNPC1ALDH1A1RAB9ATDP1
SCHEMBL7310787 0.79 TDP1 (0.55) MAPTALDH1A1TDP1KDM4ESMN1; SMN2
SCHEMBL7310781 0.79 TDP1 (0.55) MAPTALDH1A1TDP1KDM4ESMN1; SMN2
SCHEMBL7301102 0.77 ALDH1A1 (0.39) MAPTALDH1A1KDM4ESMN1; SMN2MEN1
SCHEMBL7301097 0.77 ALDH1A1 (0.39) MAPTALDH1A1KDM4ESMN1; SMN2MEN1
SCHEMBL7304760 0.76 MAPT (0.47) PKMMAPTALDH1A1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed