SCHEMBL7310787

SCHEMBL7310787

CC(C)[C@H](NC(=O)N(C)Cc1nc2ccccc2[nH]1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.55
PIN1 Q13526 4/20 0.51
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MAPT P10636 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CHRM1 P11229 1/20 0.46
BCHE P06276 1/20 0.46
HTT P42858 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310781 1.00 TDP1 (0.55) TDP1PIN1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7302465 0.89 ALDH1A1 (0.50) TDP1PIN1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7302472 0.89 ALDH1A1 (0.50) TDP1PIN1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL7333130 0.83 CA2 (0.64) TDP1PIN1ALDH1A1KDM4EMAPT
SCHEMBL7333674 0.83 CA2 (0.64) TDP1PIN1ALDH1A1KDM4EMAPT
SCHEMBL7333388 0.83 CA2 (0.64) TDP1PIN1ALDH1A1KDM4EMAPT
SCHEMBL11353994 0.80 TDP1 (0.68) TDP1ALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL7307810 0.79 PKM (0.49) TDP1ALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL7307803 0.79 PKM (0.49) TDP1ALDH1A1SMN1; SMN2KDM4EMAPT
SCHEMBL7310994 0.79 CA2 (0.67) TDP1ALDH1A1KDM4EMAPTCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed