SCHEMBL7307824

SCHEMBL7307824

Cn1c(CC2CCN(CCCNS(C)(=O)=O)CC2)c(C(=O)O)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 5/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
ALOX15 P16050 1/20 0.49
NFKB1 P19838 1/20 0.49
PMP22 Q01453 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
KCNH2 Q12809 2/20 0.46
MAPT P10636 1/20 0.44
HTR7 P34969 4/20 0.44
RAB9A P51151 1/20 0.43
CCR3 P51677 2/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A3 Q01959 1/20 0.42
CNR2 P34972 1/20 0.42
MEN1 O00255 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4294891 0.94 HTR4 (0.55) HTR4CYP1A2CYP2C9ALOX15NFKB1
Fumaric Acid SCHEMBL2942179 0.90 HTR4 (0.51) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL9704182 0.87 HTR4 (0.63) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL9341470 0.85 HTR4 (0.50) HTR4PMP22NPSR1KCNH2HTR7
SCHEMBL7308950 0.85 KDM1A (0.46) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7304868 0.83 SLC6A2 (0.47) MAPTHTR7RAB9ASLC6A2SLC6A3
SCHEMBL7300755 0.82 KDM4E (0.46) HTR4MAPTHTR7SLC6A2SLC6A3
SCHEMBL7309279 0.82 KDM1A (0.45) HTR4CYP1A2CYP2C9MAPTHTR7
SCHEMBL7304670 0.82 KDM1A (0.46) MAPTHTR7SMN1; SMN2AGTR1
SCHEMBL7303226 0.81 CYP2C9 (0.49) HTR4CYP1A2CYP2C9ALOX15NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP claimed