SCHEMBL9704182

SCHEMBL9704182

Cn1c(CC2CCN(CCNS(C)(=O)=O)CC2)c(C(=O)O)c2ccccc21.Cn1cc(C(=O)O)c2ccccc21

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 5/20 0.63
CYP1A2 P05177 1/20 0.63
CYP2C9 P11712 1/20 0.63
ALOX15 P16050 1/20 0.63
NFKB1 P19838 1/20 0.63
PMP22 Q01453 1/20 0.63
NPSR1 Q6W5P4 1/20 0.63
BCHE P06276 2/20 0.46
ACHE P22303 2/20 0.46
KCNH2 Q12809 2/20 0.46
KDM1A O60341 1/20 0.40
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4294891 0.92 HTR4 (0.55) HTR4CYP1A2CYP2C9ALOX15NFKB1
Fumaric Acid SCHEMBL2942179 0.88 HTR4 (0.51) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7307824 0.87 HTR4 (0.49) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7324773 0.86 HTR4 (0.69) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7308950 0.83 KDM1A (0.46) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7304868 0.80 SLC6A2 (0.47) SLC6A2SLC6A3
SCHEMBL7303226 0.80 CYP2C9 (0.49) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL7301718 0.79 HTR4 (0.62) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL4294889 0.78 HTR4 (0.61) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL1502039 0.78 HTR4 (1.00) HTR4CYP1A2CYP2C9ALOX15NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992014727-A1 3-PIPERIDINYLMETHYLCARBOXYLATE SUBSTITUTED INDOLES GLAXO GROUP LIMITED (GB) 1992-09-03 WO disclosed