SCHEMBL7308950

SCHEMBL7308950

Cn1c(CC2CCN(CCNS(=O)(=O)c3ccccc3)CC2)c(C(=O)O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.46
HTR4 Q13639 4/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44
PMP22 Q01453 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
KDM4E B2RXH2 2/20 0.43
KCNH2 Q12809 2/20 0.42
HTR7 P34969 2/20 0.42
SLC6A2 P23975 2/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4294891 0.90 HTR4 (0.55) KDM1AHTR4CYP1A2CYP2C9ALOX15
Fumaric Acid SCHEMBL2942179 0.86 HTR4 (0.51) KDM1AHTR4CYP1A2CYP2C9ALOX15
SCHEMBL7304868 0.85 SLC6A2 (0.47) KDM4EHTR7SLC6A2SLC6A3PRMT6
SCHEMBL7307824 0.85 HTR4 (0.49) HTR4CYP1A2CYP2C9ALOX15NFKB1
SCHEMBL9704182 0.83 HTR4 (0.63) KDM1AHTR4CYP1A2CYP2C9ALOX15
SCHEMBL7300755 0.82 KDM4E (0.46) HTR4ALDH1A1SMN1; SMN2KDM4EHTR7
SCHEMBL7309279 0.82 KDM1A (0.45) KDM1AHTR4CYP1A2CYP2C9KDM4E
SCHEMBL9341470 0.81 HTR4 (0.50) HTR4PMP22NPSR1ALDH1A1KDM4E
SCHEMBL7302843 0.80 KDM4E (0.44) HTR4NPSR1ALDH1A1MEN1KMT2A
SCHEMBL7301395 0.80 HTR7 (0.46) HTR4ALDH1A1SMN1; SMN2KDM4EHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP claimed