SCHEMBL7307892

SCHEMBL7307892

COc1cccc2c1OC(CNCC1CCCCC1)CC2

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.56
HTR1D P28221 1/20 0.56
ADRA1D P25100 7/20 0.47
ADRA1A P35348 7/20 0.47
ADRA1B P35368 7/20 0.47
HTR2C P28335 1/20 0.44
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
HPGD P15428 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317381 1.00 HTR1A (0.56) HTR1AHTR1DADRA1DADRA1AADRA1B
SCHEMBL7321215 1.00 HTR1A (0.56) HTR1AHTR1DADRA1DADRA1AADRA1B
SCHEMBL7318030 1.00 HTR1A (0.56) HTR1AHTR1DADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL467043 0.99 HTR1A (0.55) HTR1AHTR1DADRA1DADRA1AADRA1B
SCHEMBL7313874 0.87 NFKB1 (0.46) HTR1AHTR1DADRA1DADRA1AADRA1B
SCHEMBL7309189 0.83 NFKB1 (0.44) HTR1AHTR1DADRA1DADRA1AADRA1B
Cyclohexane SCHEMBL8317149 0.82 HTR1A (0.50) HTR1AHTR1DNFKB1NFKB2RELA
Cycloheptane SCHEMBL8315045 0.82 HTR1A (0.50) HTR1AHTR1DNFKB1NFKB2RELA
SCHEMBL7321928 0.82 KMT2A (0.50) HTR1AHTR1DADRA1ANFKB1NFKB2
SCHEMBL7313786 0.82 KMT2A (0.50) HTR1AHTR1DADRA1ANFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5318988-A Treating psychoses BAYER AKTIENGESELLSCHAFT (DE) 1994-06-07 US claimed
US-5962513-A CENTRAL NERVOUS SYSTEM, PSYCHOLOGICAL DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1999-10-05 US disclosed
EP-0540914-B1 2-Aminomethylchromans as active ingredients in medicaments for the treatment of diseases of the central nervous system BAYER AG (DE) 1999-06-02 EP disclosed
US-5468882-A Serotoninergic agents; central nervous system and psychological disorders BAYER AKTIENGESELLSCHAFT (DE) 1995-11-21 US disclosed
US-5318988-A Treating psychoses BAYER AKTIENGESELLSCHAFT (DE) 1994-06-07 US disclosed
EP-0540914-A1 2-Aminomethylchromans as active ingredients in medicaments for the treatment of diseases of the central nervous system BAYER AG (DE) 1993-05-12 EP disclosed