SCHEMBL730902

SCHEMBL730902

COc1c[c]cc(-c2nnn[nH]2)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
XDH P47989 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
SCN4A P35499 1/20 0.30
CYP1A1 P04798 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL732864 0.84 ALDH1A1 (0.35) ALDH1A1HPGDSMN1; SMN2HSD17B10GAA
SCHEMBL733135 0.77
SCHEMBL703677 0.75 DCUN1D1 (0.54) GAAMAPTNR1H2NR1H3XDH
SCHEMBL31357013 0.75 CYP1A1 (0.46) CYP1A1CYP1B1
SCHEMBL6744136 0.75 ALDH1A1 (0.41) ALDH1A1HPGDSMN1; SMN2HSD17B10GAA
SCHEMBL731571 0.75 NR1H2 (0.44) SMN1; SMN2MAPTNR1H2NR1H3XDH
SCHEMBL672108 0.74 KDM4E (0.50) ALDH1A1HPGDSMN1; SMN2GAAMAPT
SCHEMBL18758173 0.73 XDH (0.50) ALDH1A1HPGDSMN1; SMN2GAAMAPT
SCHEMBL731417 0.72 GP6 (0.37) ALDH1A1NR1H2NR1H3SCN4A
SCHEMBL733059 0.72 NPC1 (0.40) ALDH1A1HPGDSMN1; SMN2GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-B1 SPIROCHROMANON DERIVATIVES MERCK SHARP & DOHME (US) 2013-08-14 EP disclosed
US-8138197-B2 Spirochromanon derivatives MSD K.K. (JP) 2012-03-20 US disclosed
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
US-20090270436-A1 SPIROCHROMANON DERIVATIVES MERCK SHARP & DOHME LLC 2009-10-29 US disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090270436-A1 SPIROCHROMANON DERIVATIVES AKR1C3, CBR3, AKR1C4 ALDH1A1 113/4885HPGD 2417/4885SMN1; SMN2 3531/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.