SCHEMBL7309324

SCHEMBL7309324

CC(C)(C)ONC(=O)CC(Cc1ccccc1)Sc1cc(-c2ccccc2)cs1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.36
KLK5 Q9Y337 1/20 0.36
MMP12 P39900 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
PPARG P37231 8/20 0.34
PPARA Q07869 6/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.34
ITGA4 P13612 1/20 0.34
ITGB7 P26010 1/20 0.34
CTSB P07858 1/20 0.34
MME P08473 1/20 0.33
ACE2 Q9BYF1 1/20 0.33
MMP2 P08253 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
PSMB8 P28062 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301211 0.84 MME (0.41) MMEMMP2
SCHEMBL7301071 0.83 CTSS (0.41) ACELMNAPPARGPPARACTSS
SCHEMBL7302926 0.81 CPA1 (0.44) MMP12ALDH1A1PPARGPPARAMMP2
SCHEMBL7311029 0.80 CTSS (0.39) ACEKLK5MEN1ALDH1A1LMNA
SCHEMBL7309312 0.78 SLC6A4 (0.41) ACEKLK5LMNACTSSCTSK
SCHEMBL7308114 0.77 MMP2 (0.44) ACEKLK5MEN1ALDH1A1LMNA
SCHEMBL7310171 0.77 SIRT5 (0.44) MEN1ALDH1A1LMNAKMT2APPARG
SCHEMBL27478790 0.76 PPARG (0.48) PPARGPPARA
SCHEMBL7310105 0.75 PPARG (0.42) PPARGPPARAMMP2MMP13
SCHEMBL7304806 0.75 PPARG (0.44) ALDH1A1KMT2APPARGPPARAMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed