SCHEMBL7309366

SCHEMBL7309366

Cc1ccccc1-n1nnnc1CCCOc1ccc2[nH]c(=O)ccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.44
DRD2 P14416 8/20 0.43
DRD4 P21917 4/20 0.43
DRD3 P35462 4/20 0.43
PDE3B Q13370 5/20 0.40
PDE3A Q14432 5/20 0.40
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
MEN1 O00255 1/20 0.40
PDE5A O76074 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
PTAFR P25105 1/20 0.40
BLM P54132 1/20 0.40
PDE1A P54750 1/20 0.40
PDE1B Q01064 1/20 0.40
PMP22 Q01453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310025 0.86 PKM (0.44) HSD11B1DRD2DRD4DRD3PDE3B
SCHEMBL7307423 0.83 ALDH1A1 (0.40) DRD2DRD4DRD3PDE3BPDE3A
SCHEMBL7316070 0.83 ALDH1A1 (0.43) DRD2DRD4DRD3PDE3BPDE3A
SCHEMBL7320251 0.82 MAPT (0.48) PDE3BPDE3AKDM4EALDH1A1CYP1A2
SCHEMBL7317769 0.82 PDE3B (0.45) DRD2DRD4DRD3PDE3BPDE3A
SCHEMBL7307849 0.81 KCNH2 (0.47) DRD2PDE3BPDE3AKDM4EALDH1A1
SCHEMBL7312406 0.80 PDE3B (0.43) DRD2DRD4DRD3PDE3BPDE3A
SCHEMBL7341497 0.79 PDE3B (0.43) DRD2DRD4DRD3PDE3BPDE3A
SCHEMBL7313419 0.79 PDE3B (0.48) PDE3BPDE3AKDM4EALDH1A1CYP1A2
SCHEMBL7304090 0.79 KDM4E (0.43) DRD2DRD4DRD3PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4277479-A ANTI-ASTHMATIC, HYPOTENSIVE, ANTI-ULCER, ANTIINFLAMMATORY, VASODILATION, ENZYME INHIBITORS, ANTICOAGULANTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-07-07 US disclosed