SCHEMBL7310025

SCHEMBL7310025

O=c1ccc2cc(OCCCc3nnnn3-c3ccccc3)ccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.44
HTT P42858 1/20 0.44
NLRP3 Q96P20 1/20 0.44
ALDH1A1 P00352 7/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 1/20 0.43
PDE3B Q13370 3/20 0.42
PDE3A Q14432 3/20 0.42
HSD11B1 P28845 3/20 0.40
TSHR P16473 3/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
MCL1 Q07820 1/20 0.40
PDE5A O76074 1/20 0.40
HPGD P15428 1/20 0.40
PTAFR P25105 1/20 0.40
BLM P54132 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316070 0.90 ALDH1A1 (0.43) HTTALDH1A1KMT2ALMNAPDE3B
SCHEMBL7307849 0.90 KCNH2 (0.47) ALDH1A1KMT2ALMNAPDE3BPDE3A
SCHEMBL7309366 0.86 HSD11B1 (0.44) ALDH1A1KMT2APDE3BPDE3AHSD11B1
SCHEMBL7313419 0.84 PDE3B (0.48) PKMHTTALDH1A1KMT2ALMNA
SCHEMBL7320251 0.84 MAPT (0.48) ALDH1A1KMT2ALMNAPDE3BPDE3A
SCHEMBL7312752 0.83 HCAR1 (0.40) PKMHTTALDH1A1KMT2ALMNA
SCHEMBL7303943 0.83 ALDH1A1 (0.53) ALDH1A1KMT2ALMNAPDE3BPDE3A
SCHEMBL7317769 0.83 PDE3B (0.45) ALDH1A1KMT2ALMNAPDE3BPDE3A
SCHEMBL7316667 0.82 ALDH1A1 (0.42) PKMHTTNLRP3ALDH1A1KMT2A
SCHEMBL7314477 0.82 PPARA (0.45) PKMHTTNLRP3ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4277479-A ANTI-ASTHMATIC, HYPOTENSIVE, ANTI-ULCER, ANTIINFLAMMATORY, VASODILATION, ENZYME INHIBITORS, ANTICOAGULANTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-07-07 US claimed
US-4277479-A ANTI-ASTHMATIC, HYPOTENSIVE, ANTI-ULCER, ANTIINFLAMMATORY, VASODILATION, ENZYME INHIBITORS, ANTICOAGULANTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-07-07 US disclosed