SCHEMBL7309877

SCHEMBL7309877

O=C1C(CN2CCN(CCCO)CC2)CCN1c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.46
HTR1A P08908 2/20 0.46
HTR2A P28223 2/20 0.46
HTR7 P34969 1/20 0.46
HTR6 P50406 1/20 0.46
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
DRD4 P21917 6/20 0.39
DRD3 P35462 3/20 0.39
CHRNA7 P36544 1/20 0.39
CACNA1G O43497 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
DRD1 P21728 1/20 0.38
SLC6A2 P23975 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314254 0.85 DRD2 (0.43) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL7305622 0.82 HTR2A (0.41) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL466933 0.82 KMT2A (0.44) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL466934 0.82 KMT2A (0.44) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL7315071 0.82 KMT2A (0.44) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL467338 0.82 CHRNA7 (0.52) DRD2ALDH1A1DRD3CHRNA7KDM4E
Hydrochloric Acid SCHEMBL8419734 0.81 KMT2A (0.43) DRD2HTR1AHTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL7311725 0.81 KMT2A (0.43) DRD2HTR1AHTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL467146 0.81 KMT2A (0.43) DRD2HTR1AHTR2AHTR7HTR6
Hydrochloric Acid SCHEMBL467145 0.81 KMT2A (0.43) DRD2HTR1AHTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839805-B1 Pyrrolidinone derivatives and their use as antipsychotic medicaments SCHERING AG (DE) 2001-10-04 EP disclosed
US-5969138-A ANTIPSYCHOTIC AGENTS MITSUI CHEMICALS, INC. (JP) 1999-10-19 US disclosed
EP-0839805-A1 Pyrrolidinone derivatives and their use as antipsychotic medicaments MITSUI TOATSU CHEMICALS, INC. (JP) 1998-05-06 EP disclosed