SCHEMBL466934

SCHEMBL466934

COCCN1CCN(C[C@H]2CCN(c3ccc(Cl)cc3)C2=O)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
HTR2C P28335 11/20 0.41
CHRNA7 P36544 1/20 0.40
HTR2A P28223 8/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
HTR7 P34969 1/20 0.40
HTR6 P50406 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HTR2B P41595 5/20 0.40
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
ADORA2B P29275 1/20 0.39
HTR4 Q13639 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL466933 1.00 KMT2A (0.44) KMT2AHTR2CCHRNA7HTR2AHTR1A
SCHEMBL7315071 1.00 KMT2A (0.44) KMT2AHTR2CCHRNA7HTR2AHTR1A
Hydrochloric Acid SCHEMBL467145 0.99 KMT2A (0.43) KMT2AHTR2CCHRNA7HTR2AHTR1A
Hydrochloric Acid SCHEMBL8419734 0.99 KMT2A (0.43) KMT2AHTR2CCHRNA7HTR2AHTR1A
Hydrochloric Acid SCHEMBL467146 0.99 KMT2A (0.43) KMT2AHTR2CCHRNA7HTR2AHTR1A
Hydrochloric Acid SCHEMBL7311725 0.99 KMT2A (0.43) KMT2AHTR2CCHRNA7HTR2AHTR1A
Sulfuric Acid SCHEMBL7308241 0.94 KMT2A (0.43) KMT2AHTR2CCHRNA7HTR2AHTR1A
Sulfuric Acid SCHEMBL7308229 0.94 KMT2A (0.43) KMT2AHTR2CCHRNA7HTR2AHTR1A
SCHEMBL7314254 0.93 DRD2 (0.43) CHRNA7HTR2AHTR1ADRD2HTR7
SCHEMBL7309602 0.89 HTR1A (0.41) KMT2AHTR2CHTR1ADRD2HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025233557-A1 SIGMA-1 RECEPTOR INHIBITING AGENTS FOR TREATING RHEUMATOID ARTHRITIS UNIVERSIDAD DE GRANADA (ES) 2025-11-13 WO claimed
US-6436938-B1 ADMINISTERING A SIGMA RECEPTOR LIGAND IN COMBINATION WITH AN ANTIDEPRESSANT AGENT; ESPECIALLY FOR REFRACTORY DEPRESSION PFIZER INC. 2002-08-20 US claimed
US-20020099045-A1 Combination treatment for depression PFIZER PRODUCTS INC. 2002-07-25 US claimed
EP-1224930-A1 Combination of a SR inhibitor and sigma receptor ligand in the treatment ofdepression Pfizer Products Inc. (US) 2002-07-24 EP claimed
WO-2025233557-A1 SIGMA-1 RECEPTOR INHIBITING AGENTS FOR TREATING RHEUMATOID ARTHRITIS UNIVERSIDAD DE GRANADA (ES) 2025-11-13 WO disclosed
US-20240315989-A1 METHODS OF TREATING COVID-19 WASHINGTON UNIVERSITY 2024-09-26 US disclosed
US-20240074995-A1 METHODS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH AN ABNORMAL INFLAMMATORY RESPONSES FIRST WAVE BIO, INC. 2024-03-07 US disclosed
US-11793777-B2 Methods and compositions for treating conditions associated with an abnormal inflammatory response FIRST WAVE BIO, INC. (US) 2023-10-24 US disclosed
US-11744812-B2 Methods of treatment FIRST WAVE BIO, INC. (US) 2023-09-05 US disclosed
US-20230201143-A1 METHODS OF TREATMENT FIRST WAVE BIO, INC. 2023-06-29 US disclosed
US-20230190870-A1 Method for Treating Lysosomal Storage Diseases with Histatin Peptides NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-06-22 US disclosed
US-20230102999-A1 DEUTERATED NICLOSAMIDE FIRST WAVE BIO, INC. 2023-03-30 US disclosed
EP-2415471-A1 Use of sigma ligands in opioid-induced hyperalgesia Laboratorios Del. Dr. Esteve, S.A. (ES) 2012-02-08 EP disclosed
EP-2388005-A1 Sigma ligands for the prevention and/or treatment of emesis induced by chemotherapy or radiotherapy Laboratorios Del. Dr. Esteve, S.A. (ES) 2011-11-23 EP disclosed
EP-2353598-A1 Sigma ligands for use in the prevention and/or treatment of postoperative pain Laboratorios Del. Dr. Esteve, S.A. (ES) 2011-08-10 EP disclosed
US-6436938-B1 ADMINISTERING A SIGMA RECEPTOR LIGAND IN COMBINATION WITH AN ANTIDEPRESSANT AGENT; ESPECIALLY FOR REFRACTORY DEPRESSION PFIZER INC. 2002-08-20 US disclosed
EP-1224930-A1 Combination of a SR inhibitor and sigma receptor ligand in the treatment ofdepression Pfizer Products Inc. (US) 2002-07-24 EP disclosed
EP-0839805-B1 Pyrrolidinone derivatives and their use as antipsychotic medicaments SCHERING AG (DE) 2001-10-04 EP disclosed
US-5969138-A ANTIPSYCHOTIC AGENTS MITSUI CHEMICALS, INC. (JP) 1999-10-19 US disclosed
EP-0839805-A1 Pyrrolidinone derivatives and their use as antipsychotic medicaments MITSUI TOATSU CHEMICALS, INC. (JP) 1998-05-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240074995-A1 METHODS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH AN ABNORMAL INFLAMMATORY RESPONSES FH, CS, ECHS1 KMT2A 3595/4885HTR2C 2729/4885CHRNA7 1026/4885
US-11744812-B2 Methods of treatment ACE2, ACE, SI KMT2A 2952/4885HTR2C 771/4885CHRNA7 558/4885
US-20230201143-A1 METHODS OF TREATMENT ACE2, ACE, SI KMT2A 2890/4885HTR2C 1216/4885CHRNA7 829/4885
US-20020099045-A1 Combination treatment for depression HTR5A, HTR1A, OPRL1 KMT2A 3616/4885HTR2C 10/4885CHRNA7 47/4885
US-20230102999-A1 DEUTERATED NICLOSAMIDE FH, IDH2, ECHS1 KMT2A 2551/4885HTR2C 1921/4885CHRNA7 692/4885
US-20240315989-A1 METHODS OF TREATING COVID-19 SIGMAR1, HTR1A, SGMS1 KMT2A 1259/4885HTR2C 66/4885CHRNA7 266/4885
US-11793777-B2 Methods and compositions for treating conditions associated with an abnormal inflammatory response FH, CS, ECHS1 KMT2A 3704/4885HTR2C 2736/4885CHRNA7 1162/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.