SCHEMBL7309931

SCHEMBL7309931

N#Cc1nn(C2CCCC2)c2nc(-c3ccncc3)nc(N)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.37
PIK3CD O00329 7/20 0.36
PIK3CA P42336 6/20 0.36
PIK3CB P42338 6/20 0.36
PIK3CG P48736 6/20 0.36
PRKDC P78527 6/20 0.36
ABL1 P00519 5/20 0.36
EGFR P00533 5/20 0.36
HCK P08631 5/20 0.36
SRC P12931 5/20 0.36
MTOR P42345 5/20 0.36
EPHB4 P54760 5/20 0.36
KDR P35968 4/20 0.36
RET P07949 1/20 0.36
CTSK P43235 5/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GLA P06280 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310219 0.82 PIK3CD (0.38) S1PR1PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL7315963 0.82 PIK3CD (0.38) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL7316083 0.81 KDM4E (0.46) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL7312205 0.78 PIK3CD (0.35) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL7310653 0.72 PIK3CA (0.46) S1PR1PIK3CDPIK3CAPIK3CGMTOR
SCHEMBL7308816 0.70 KDR (0.39) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL7319490 0.67 MEN1 (0.46) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL863767 0.67 RET (0.44) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL7317680 0.66 SRC (0.38) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL7312745 0.66 HPGD (0.45) ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541187-A HYPOTENSIVE AGENTS STERLING WINTHROP INC. (US) 1996-07-30 US disclosed
US-5294612-A Hypotensive agents and cardiovascular disorders STERLING WINTHROP INC. (US) 1994-03-15 US disclosed