SCHEMBL7310993

SCHEMBL7310993

COC(CCC=O)(c1ccccc1)C(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.34
CYP1A2 P05177 1/20 0.34
KCNH2 Q12809 4/20 0.34
OPRM1 P35372 2/20 0.34
OPRD1 P41143 2/20 0.34
CHRM3 P20309 2/20 0.34
MRGPRX2 Q96LB1 1/20 0.34
HRH2 P25021 1/20 0.34
HTR2A P28223 1/20 0.34
ADRA1A P35348 1/20 0.34
OPRK1 P41145 1/20 0.34
CES1 P23141 1/20 0.33
KIF11 P52732 4/20 0.33
AOX1 Q06278 1/20 0.33
LMNA P02545 2/20 0.33
KCNN4 O15554 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
RIPK1 Q13546 2/20 0.32
ALDH1A1 P00352 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819750 0.78 KCNH2 (0.35) CYP2D6CYP1A2KCNH2OPRM1OPRD1
SCHEMBL27360229 0.76 KCNN4 (0.40) KCNH2CES1KIF11AOX1LMNA
SCHEMBL21401129 0.75 KCNH2 (0.38) CYP2D6CYP1A2KCNH2OPRM1OPRD1
SCHEMBL7306462 0.75 KIF11 (0.36) CYP2D6CYP1A2KCNH2OPRM1OPRD1
SCHEMBL7307298 0.75 CYP1A2 (0.33) CYP2D6CYP1A2KIF11AOX1LMNA
SCHEMBL7307357 0.73 ALDH1A1 (0.42) CYP2D6CYP1A2KCNH2OPRM1OPRD1
SCHEMBL5752959 0.70 EBP (0.51) CYP2D6CYP1A2KCNH2OPRM1CHRM3
SCHEMBL7310593 0.70 EBP (0.51) CYP2D6CYP1A2KCNH2OPRM1CHRM3
SCHEMBL1834441 0.70 TAAR1 (0.48) OPRM1AOX1CYP2C19HIF1ARIPK1
SCHEMBL9340362 0.70 CYP2C19 (0.39) CYP2D6CYP1A2AOX1KCNN4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed