SCHEMBL7306462

SCHEMBL7306462

COC(CCCO)(c1ccccc1)C(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.36
KCNH2 Q12809 3/20 0.36
CYP2D6 P10635 2/20 0.35
CYP1A2 P05177 1/20 0.35
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
MRGPRX2 Q96LB1 1/20 0.35
CHRM3 P20309 1/20 0.35
HRH2 P25021 1/20 0.35
HTR2A P28223 1/20 0.35
ADRA1A P35348 1/20 0.35
OPRK1 P41145 1/20 0.35
CES1 P23141 1/20 0.34
ALDH1A1 P00352 3/20 0.33
CYP2C19 P33261 2/20 0.33
KCNN4 O15554 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28819750 0.79 KCNH2 (0.35) KIF11KCNH2CYP2D6CYP1A2OPRM1
SCHEMBL21401129 0.77 KCNH2 (0.38) KIF11KCNH2CYP2D6CYP1A2OPRM1
SCHEMBL7310993 0.75 CYP2D6 (0.34) KIF11KCNH2CYP2D6CYP1A2OPRM1
SCHEMBL9261644 0.72 OPRM1 (0.36) KIF11KCNH2CYP1A2OPRM1CHRM3
SCHEMBL6551716 0.72 KIF11 (0.61) KIF11KCNH2CYP2D6CHRM3CYP2C19
SCHEMBL4433640 0.72 ALDH1A1 (0.37) KIF11CYP2D6CYP1A2OPRM1CHRM3
SCHEMBL7307357 0.71 ALDH1A1 (0.42) KIF11KCNH2CYP2D6CYP1A2OPRM1
SCHEMBL27290911 0.70 LMNA (0.39) CYP2D6CYP1A2OPRM1CHRM3ALDH1A1
SCHEMBL8612132 0.70 LMNA (0.39) CYP2D6CYP1A2OPRM1CHRM3ALDH1A1
SCHEMBL7453762 0.70 KIF11 (0.59) KIF11KCNH2CYP2D6CHRM3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed