SCHEMBL7312748

SCHEMBL7312748

CCC(c1ccc(Cl)c(Cl)c1)N1CCCCC1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.68
SLC6A3 Q01959 11/20 0.68
SLC6A4 P31645 10/20 0.68
TACR1 P25103 3/20 0.43
KCNQ2 O43526 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
ADAM17 P78536 1/20 0.42
KMT2A Q03164 1/20 0.42
MCL1 Q07820 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6206712 0.82 SLC6A2 (0.62) SLC6A2SLC6A3SLC6A4TACR1SMN1; SMN2
SCHEMBL14775500 0.81 SLC6A2 (1.00) SLC6A2SLC6A3SLC6A4TACR1HRH3
SCHEMBL14775419 0.80 SLC6A2 (1.00) SLC6A2SLC6A3SLC6A4HRH3
SCHEMBL14775283 0.79 SLC6A2 (1.00) SLC6A2SLC6A3SLC6A4TACR1HRH3
Hydrochloric Acid SCHEMBL8665660 0.78 OPRM1 (0.48) SLC6A2SLC6A3SLC6A4TACR1KCNQ2
SCHEMBL10399500 0.78 SLC6A3 (0.58) SLC6A2SLC6A3SLC6A4TACR1SMN1; SMN2
SCHEMBL29585404 0.78 SLC6A3 (0.56) SLC6A2SLC6A3SLC6A4SMN1; SMN2POLB
SCHEMBL29585835 0.78 SLC6A3 (0.56) SLC6A2SLC6A3SLC6A4SMN1; SMN2POLB
SCHEMBL22206766 0.78 SLC6A3 (0.56) SLC6A2SLC6A3SLC6A4SMN1; SMN2POLB
SCHEMBL22206745 0.78 SLC6A3 (0.56) SLC6A2SLC6A3SLC6A4SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021030335-A1 A STEREOISOMERICALLY PURE NK-3 RECEPTOR ANTAGONIST AND CRYSTALLINE FORMS THEREOF MILLENDO THERAPEUTICS, INC. (US) 2021-02-18 WO disclosed
EP-0673928-B1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI SYNTHELABO (FR) 2001-08-29 EP disclosed
CN-1056605-C Compounds as selective antagonists of human tachykinin III receptor and uses thereof SANOFI CORP (FR) 2000-09-20 CN disclosed
CN-1128756-A Compounds as selective antagonists of the human tachykinin III receptor and uses thereof SANOFI CORP (FR) 1996-08-14 CN disclosed
EP-0673928-A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI (FR) 1995-09-27 EP disclosed
EP-0673928-A1 Novel N-(3,4-dichlorophenyl-propyl)-piperidine derivatives as selective human NK3-receptor antagonists SANOFI (FR) 1995-09-27 EP disclosed